Pitofenone hydrochloride

CAS No. 1248-42-6

Pitofenone hydrochloride( Pitofenone hydrochloride | Pitofenone HCl | Bulgarketone )

Catalog No. M17905 CAS No. 1248-42-6

Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.

Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 35 In Stock
10MG 65 In Stock
25MG 147 In Stock
50MG 281 In Stock
100MG 528 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    Pitofenone hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
  • Description
    Pitofenone hydrochloride is an antispasmodic agent. It acts as a potent inhibitor of acetylcholinesterase activity.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Pitofenone hydrochloride | Pitofenone HCl | Bulgarketone
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    AChE
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1248-42-6
  • Formula Weight
    403.9
  • Molecular Formula
    C22H26ClNO4
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 103.3 mg/mL 255.76 mM;
  • SMILES
    Cl.O=C(OC)c1ccccc1C(=O)c3ccc(OCCN2CCCCC2)cc3
  • Chemical Name
    Methyl 2-[4-(2-piperidin-1-ylethoxy)benzoyl]benzoate hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Punekar NS,etal.Acetylcholinesterase inhibition by pitofenone: a spasmolytic compound.Biotechnol Appl Biochem. 1991 Dec;14(3):378-82.
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