Pitofenone hydrochloride

CAS No. 1248-42-6

Pitofenone hydrochloride ( Pitofenone hydrochloride; Pitofenone HCl;Bulgarketone )

Catalog No. M17905 CAS No. 1248-42-6

Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 65 In Stock
25MG 147 In Stock
50MG 281 In Stock
100MG 528 In Stock
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Biological Information

  • Product Name
    Pitofenone hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
  • Description
    Pitofenone hydrochloride is an antispasmodic agent. It acts as a potent inhibitor of acetylcholinesterase activity.
  • Synonyms
    Pitofenone hydrochloride; Pitofenone HCl;Bulgarketone
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    AChE
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1248-42-6
  • Formula Weight
    403.9
  • Molecular Formula
    C22H26ClNO4
  • Purity
    98%
  • Solubility
    DMSO : 103.3 mg/mL 255.76 mM;
  • SMILES
    Cl.O=C(OC)c1ccccc1C(=O)c3ccc(OCCN2CCCCC2)cc3
  • Chemical Name
    Methyl 2-[4-(2-piperidin-1-ylethoxy)benzoyl]benzoate hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Punekar NS,etal.Acetylcholinesterase inhibition by pitofenone: a spasmolytic compound.Biotechnol Appl Biochem. 1991 Dec;14(3):378-82.
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