Pitofenone hydrochloride
CAS No. 1248-42-6
Pitofenone hydrochloride( Pitofenone hydrochloride | Pitofenone HCl | Bulgarketone )
Catalog No. M17905 CAS No. 1248-42-6
Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
Purity : >98% (HPLC)
Size | Price / USD | Stock | Quantity |
5MG | 35 | In Stock |
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10MG | 65 | In Stock |
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25MG | 147 | In Stock |
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50MG | 281 | In Stock |
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100MG | 528 | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NamePitofenone hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionPitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
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DescriptionPitofenone hydrochloride is an antispasmodic agent. It acts as a potent inhibitor of acetylcholinesterase activity.
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In Vitro——
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In Vivo——
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SynonymsPitofenone hydrochloride | Pitofenone HCl | Bulgarketone
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PathwayOthers
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TargetOther Targets
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RecptorAChE
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Research Area——
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Indication——
Chemical Information
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CAS Number1248-42-6
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Formula Weight403.9
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Molecular FormulaC22H26ClNO4
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Purity>98% (HPLC)
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SolubilityDMSO : 103.3 mg/mL 255.76 mM;
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SMILESCl.O=C(OC)c1ccccc1C(=O)c3ccc(OCCN2CCCCC2)cc3
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Chemical NameMethyl 2-[4-(2-piperidin-1-ylethoxy)benzoyl]benzoate hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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R715 TFA(185052-09-9...
Potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Metabolically stable.
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α-Hydroxyisobutyric ...
Alpha-Hydroxyisobutyric acid is a metabolite of methyl tert-butyl ether (MTBE). MTBE may be obtained through environmental exposure. MTBE is rapidly eliminated from the body mainly through expired air as the unchanged compound. MTBE is to some extent metabolised to t-butyl alcohol (TBA) and formaldehyde and oxidised to 2-methyl-12-propanediol and a-hydroxy isobuturic acid. Alpha-Hydroxyisobutyric acid has been used as an arial bactericide.
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Isofutoquinol A
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